The development of glycosylation methods is reviewed.Numberous methods are roughly classified into 7 groups based on their type of anomeric functional group and the reaction path of glycosylation.

• 本文重点介绍了低聚糖合成的各种方法，评述了糖苷化反应的各种新进展以及存在的问题，并根据其不同的特点进行了分类。