Six 3-aryloxy-1-propylamines were synthesized for studying the SAR of HIV-1 Tat/PCAF BRD inhibitors.

• 测定结果进一步补充完善了N_1-(芳基)-(CH_2)_n-二胺盐酸盐类小分子化学抑制剂的构效关系(SAR)。