It was confirmed that the synthesis of lipoylbenzotriazole was successful by its modification reaction with insulin, and lipoylbenzotriazole showed a high reaction activity as an acylating agent.

• 通过考察硫辛酰苯并三唑对胰岛素的化学修饰作用，进一步证明了它的合成是成功的，并且对胰岛素的侧链氨基呈现较高的修饰反应活性。