As leading compounds these stilenes were modified by alkylation, glycosylation and association on the basis of the theory of structure modification and the theory of structure-activity relationships.

• 对取代苯甲醛和取代苯乙腈分别进行糖基化修饰,通过相转移催化法合成相应的糖苷中间体,后者经缩合得到糖基化修饰产物。